SCHEMBL416478

SCHEMBL416478

Cc1cccc(-c2nnc(C)[nH]2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I3 Q14994 1/20 0.50
PIN1 Q13526 1/20 0.47
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46
NPBWR1 P48145 1/20 0.44
TYMP P19971 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
IDO1 P14902 1/20 0.43
METAP2 P50579 1/20 0.43
PBRM1 Q86U86 1/20 0.43
NPY5R Q15761 1/20 0.43
MAPK14 Q16539 1/20 0.43
ALDH1A1 P00352 2/20 0.42
NISCH Q9Y2I1 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
XDH P47989 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL416660 0.81 GAA (0.53) PIN1NPBWR1TYMPIDO1NPY5R
SCHEMBL1077128 0.81 NPC1 (0.51) RAB9ANPC1HPGDTSHRSMN1; SMN2
SCHEMBL17713903 0.81 PIN1 (0.45) NR1I3PIN1RAB9ANPC1NPBWR1
Water SCHEMBL17103297 0.80 NPC1 (0.50) RAB9ANPC1HPGDTSHRSMN1; SMN2
SCHEMBL416435 0.79 POLB (0.60) PIN1RAB9ANPC1HPGDSMN1; SMN2
SCHEMBL22307332 0.79 PIN1 (0.43) NR1I3PIN1RAB9ANPC1NPBWR1
SCHEMBL416539 0.79 CYP1A2 (0.52) NR1I3PIN1TYMPNPY5RMAPK14
SCHEMBL15330749 0.78 PIN1 (0.46) NR1I3PIN1RAB9ANPC1NPBWR1
SCHEMBL19559083 0.76 NPC1 (0.54) PIN1RAB9ANPC1HPGDTSHR
SCHEMBL417398 0.76 DHODH (0.47) NR1I3PIN1NPC1HPGDMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US claimed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US claimed
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US disclosed
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US disclosed
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2012-01-26 US disclosed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US disclosed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US disclosed
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION ADHEREX TECHNOLOGIES, INC. (CA) 2009-11-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090291967-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION CDH1, EPCAM, ICAM1 NR1I3 1963/4885PIN1 3264/4885RAB9A 100/4885
US-20120022083-A1 SMALL MOLECULE MODULATORS OF CELL ADHESION CDH1, EPCAM, ICAM1 NR1I3 1963/4885PIN1 3264/4885RAB9A 100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.