SCHEMBL4171179

SCHEMBL4171179

C=CCc1cc[nH]c1C=O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
POLB P06746 1/20 0.33
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27686311 0.83 GABRA1 (0.35) GABRA1GABRB2POLB
SCHEMBL4053225 0.79
SCHEMBL11441284 0.78 GABRA1 (0.41) GABRA1GABRB2KDM4E
SCHEMBL1491968 0.75
SCHEMBL8718496 0.74 GABRA1 (0.48) GABRA1GABRB2POLBKDM4E
SCHEMBL27835308 0.73
SCHEMBL1655686 0.72 GABRA1 (0.36) GABRA1GABRB2POLB
SCHEMBL7613712 0.72 CHEK1 (0.37)
SCHEMBL14560346 0.72 SRC (0.43) GABRA1GABRB2POLBKDM4E
SCHEMBL9225445 0.72 GPR84 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683546-A Alkyl pyrrole aldehyde derivative and preparation method and application thereof 厦门医学院 2021-11-23 CN disclosed
CN-113683546-A Alkyl pyrrole aldehyde derivative and preparation method and application thereof 厦门医学院 2021-11-23 CN disclosed
CN-109467558-B 1-hydropyrrolizine derivative and synthesis method and application thereof 广西师范大学 2021-03-23 CN disclosed
WO-2009084007-A1 PYRROLE END-CAPPED BIPYRIDINE ASSAY POWDER FOR SELECTIVE DETECTION OF ZINC IONS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-07-09 WO disclosed
US-6441194-B1 TWO STEP, ONE POT ALKYLATION IN PRESENCE OF BRONSTEAD ACID CATALYST; REACTING PYRROLE-2-CARBALDEHYDE WITH VILSMEIR REAGENT, SUCH AS OXALYL CHLORIDE AND DIMETHYLFORAMIDE, THEN ALKYLATING AGENT, SUCH AS TERTBUTYL CHORIDE EMORY UNIVERSITY 2002-08-27 US disclosed
WO-2001028997-A2 SYNTHESIS OF 4-SUBSTITUTED PYRROLE-2-CARBALDEHYDE COMPOUNDS EMORY UNIVERSITY (US) 2001-04-26 WO disclosed