SCHEMBL4178157

SCHEMBL4178157

CC(C)(C)OC(=O)n1c(Cn2c(CN3CCC4CCc5cccnc5C43)nc3ccccc32)nc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 1/20 0.39
NOD1 Q9Y239 1/20 0.39
CXCR4 P61073 9/20 0.36
GPR119 Q8TDV5 2/20 0.36
FNTA P49354 3/20 0.35
FNTB P49356 3/20 0.35
CYP2D6 P10635 1/20 0.34
MMP3 P08254 1/20 0.33
MMP7 P09237 1/20 0.33
MMP10 P09238 1/20 0.33
MMP8 P22894 1/20 0.33
MMP12 P39900 1/20 0.33
ALDH1A2 O94788 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ALDH2 P05091 2/20 0.33
ALDH3A1 P30838 2/20 0.33
ALDH1A3 P47895 2/20 0.33
OPRL1 P41146 2/20 0.33
KCNH2 Q12809 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13875272 1.00 NOD2 (0.39) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL4163663 0.96 GPR119 (0.38) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL13875271 0.96 GPR119 (0.38) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL13875189 0.91 CXCR4 (0.41) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL4171449 0.91 CXCR4 (0.41) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL4185850 0.91 CXCR4 (0.41) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL4171448 0.91 CXCR4 (0.41) NOD2NOD1CXCR4GPR119FNTA
SCHEMBL13875254 0.82 CXCR4 (0.45) NOD2NOD1CXCR4FNTAFNTB
SCHEMBL4179325 0.78 CXCR4 (0.51) CXCR4FNTAFNTBCYP2D6KCNH2
SCHEMBL13875218 0.78 CXCR4 (0.51) CXCR4FNTAFNTBCYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090093454-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2009-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090093454-A1 Chemical Compounds SLC10A1, CYP11B2, CYP4F3 NOD2 2852/4885NOD1 2562/4885CXCR4 2681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.