SCHEMBL4181668

SCHEMBL4181668

CCOC(=O)c1nn(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)c1CO

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
CA4 P22748 1/20 0.55
CA9 Q16790 1/20 0.55
KMT2A Q03164 1/20 0.53
KDM4E B2RXH2 1/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
ALDH1A1 P00352 3/20 0.51
GABRA2 P47869 2/20 0.51
GABRB2 P47870 2/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MAPT P10636 3/20 0.50
LMNA P02545 1/20 0.50
APP P05067 1/20 0.50
CASP1 P29466 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
CYP19A1 P11511 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4186603 0.89 CA1 (0.54) CA1CA2CA4CA9KMT2A
SCHEMBL4187519 0.86 CA1 (0.58) CA1CA2CA4CA9KMT2A
SCHEMBL4193262 0.85 CNR1 (0.60) GABRA2GABRB2
SCHEMBL4184217 0.85 CNR1 (0.53) CYP19A1
SCHEMBL29838942 0.81 ALDH1A1 (0.63) CA1CA2CA4CA9KMT2A
SCHEMBL12053889 0.80 CNR1 (0.62) GABRA2GABRB2
SCHEMBL4914356 0.80 GABRA2 (0.60) KMT2AKDM4EGABRA2GABRB2MAPT
SCHEMBL277032 0.79 KDM4E (0.51) CA1CA2CA4CA9KMT2A
SCHEMBL276776 0.78 CNR1 (0.57) CA1CA2CA4CA9KMT2A
SCHEMBL4872470 0.78 GABRA2 (0.59) CA1CA2CA4CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095752-A1 FUSED PYRAZOLE DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-08-06 WO disclosed