SCHEMBL4187519

SCHEMBL4187519

CCOC(=O)c1nn(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)c1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA4 P22748 1/20 0.58
CA9 Q16790 1/20 0.58
CNR1 P21554 2/20 0.57
KMT2A Q03164 1/20 0.56
KDM4E B2RXH2 1/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
GABRA2 P47869 1/20 0.54
GABRB2 P47870 1/20 0.54
ALDH1A1 P00352 2/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
APP P05067 1/20 0.53
MAPT P10636 1/20 0.53
CASP1 P29466 1/20 0.53
CYP19A1 P11511 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29838942 0.94 ALDH1A1 (0.63) CA1CA2CA4CA9CNR1
SCHEMBL277032 0.91 KDM4E (0.51) CA1CA2CA4CA9CNR1
SCHEMBL4872470 0.91 GABRA2 (0.59) CA1CA2CA4CA9CNR1
SCHEMBL276776 0.88 CNR1 (0.57) CA1CA2CA4CA9CNR1
SCHEMBL327857 0.88 CNR1 (0.53) CA1CA2CA4CA9CNR1
SCHEMBL276777 0.87 CNR1 (0.54) CA1CA2CA4CA9CNR1
SCHEMBL4181668 0.86 CA1 (0.55) CA1CA2CA4CA9KMT2A
SCHEMBL4186603 0.85 CA1 (0.54) CA1CA2CA4CA9KMT2A
SCHEMBL29838956 0.84 CNR2 (0.71) CNR1CNR2
SCHEMBL700719 0.84 CNR1 (0.58) CNR1CYP19A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095752-A1 FUSED PYRAZOLE DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-08-06 WO disclosed