SCHEMBL4183383

SCHEMBL4183383

Cc1ccc(C(=O)N2CCC(O)(c3ccc(C(F)(F)F)cc3)CC2)cc1NS(C)(=O)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.44
EPHX2 P34913 1/20 0.44
KDM4E B2RXH2 1/20 0.43
PKLR P30613 2/20 0.43
CA12 O43570 3/20 0.42
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA7 P43166 3/20 0.42
CA9 Q16790 3/20 0.42
CA14 Q9ULX7 3/20 0.42
S1PR2 O95136 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KDM1A O60341 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
DRD2 P14416 1/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
FASN P49327 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4186712 0.90 PKLR (0.55) KDM4EPKLRALDH1A1SMN1; SMN2MEN1
SCHEMBL4172413 0.87 KDM4E (0.58) KDM4EPKLRCA12CA1CA2
SCHEMBL4172798 0.87 CA12 (0.57) KDM4EPKLRCA12CA1CA2
SCHEMBL4181151 0.87 CA12 (0.56) KDM4EPKLRCA12CA1CA2
SCHEMBL4174590 0.81 FASN (0.56) FASNGAA
SCHEMBL4187265 0.80 PKLR (0.52) PKLR
SCHEMBL29844006 0.75 MEN1 (0.55) CYP2C9EPHX2CA12CA1CA2
SCHEMBL4177346 0.73 CA12 (0.50) KDM4EPKLRCA12CA1CA2
SCHEMBL4203520 0.72 MEN1 (0.49) CYP2C9KDM4EPKLRSMN1; SMN2MEN1
SCHEMBL4182807 0.72 FASN (0.51) PKLRFASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090105305-A1 Therapeutic Agents - 550 ASTRAZENECA AB (SE) 2009-04-23 US disclosed
WO-2008075070-A1 SULFONAMIDE DERIVATIVES FOR THERAPEUTIC USE AS FATTY ACID SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090105305-A1 Therapeutic Agents - 550 FABP4, GPR119, FASN CYP2C9 3068/4885EPHX2 1986/4885KDM4E 2575/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.