SCHEMBL4184836

SCHEMBL4184836

CCCCCn1c(=O)n(C)c2cnc(Cl)nc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 10/20 0.43
ADORA2A P29274 9/20 0.43
PDE4B Q07343 9/20 0.43
PDE4C Q08493 9/20 0.43
PDE4D Q08499 9/20 0.43
ADORA2B P29275 4/20 0.43
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41
TNF P01375 1/20 0.40
LMNA P02545 4/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TSHR P16473 1/20 0.37
NR2F2 P24468 1/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20367292 0.84 TRPC5 (0.35) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL30328166 0.78 HPGD (0.38) HTTHPGDHSD17B10
SCHEMBL23620552 0.77 HPGD (0.56) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL1693503 0.77 HPGD (0.54) ADORA2BTP53HTTHPGDHSD17B10
SCHEMBL30031420 0.76 PIK3CA (0.46) LMNAPOLBHTTHSD17B10TSHR
SCHEMBL7504710 0.75 CDK4 (0.56)
SCHEMBL28682158 0.75 TSHR (0.40) ADORA2ALMNAPOLBHPGDTSHR
SCHEMBL29351994 0.75 TSHR (0.40) ADORA2ALMNAPOLBHPGDTSHR
SCHEMBL4191402 0.74 PDE4A (0.45) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL24572009 0.74 HSD17B10 (0.37) ADORA2ALMNAHTTHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029145-A2 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES Novartis Ag (CH) 2009-03-04 EP disclosed
WO-2007140222-A2 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2007-12-06 WO disclosed