SCHEMBL4189374

SCHEMBL4189374

COc1cc(/C=C(\C#N)S(=O)(=O)Cc2ccc(F)cc2)cc(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 4/20 0.47
PTGS1 P23219 1/20 0.45
PKM P14618 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HPGD P15428 1/20 0.42
EGFR P00533 3/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ERBB2 P04626 1/20 0.39
PTPN7 P35236 1/20 0.38
PTPN12 Q05209 1/20 0.38
PTPN22 Q9Y2R2 1/20 0.38
KIF20A O95235 1/20 0.37
MAOB P27338 1/20 0.37
CYP24A1 Q07973 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4189380 1.00 NQO2 (0.47) NQO2PTGS1PKML3MBTL1HPGD
SCHEMBL4189377 1.00 NQO2 (0.47) NQO2PTGS1PKML3MBTL1HPGD
SCHEMBL4192011 0.91 NQO2 (0.53) NQO2PTGS1PKMHPGDEGFR
SCHEMBL4192017 0.91 NQO2 (0.53) NQO2PTGS1PKMHPGDEGFR
SCHEMBL4192014 0.91 NQO2 (0.53) NQO2PTGS1PKMHPGDEGFR
SCHEMBL4168075 0.89 PKM (0.54) PKML3MBTL1HPGDEGFRMEN1
SCHEMBL4184666 0.89 ALDH1A1 (0.46) NQO2PKML3MBTL1HPGDEGFR
SCHEMBL4184669 0.89 ALDH1A1 (0.46) NQO2PKML3MBTL1HPGDEGFR
SCHEMBL4184673 0.89 ALDH1A1 (0.46) NQO2PKML3MBTL1HPGDEGFR
SCHEMBL4168077 0.89 PKM (0.54) PKML3MBTL1HPGDEGFRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090191193-A1 Aryl Vinyl Sulfides, Sulfones, Sulfoxides and Sulfonamides, Derivatives Thereof and Therapeutic Uses Thereof TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-07-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090191193-A1 Aryl Vinyl Sulfides, Sulfones, Sulfoxides and Sulfonamides, Derivatives Thereof and Therapeutic Uses Thereof ARSA, STS, SULT2A1 NQO2 1049/4885PTGS1 741/4885PKM 2657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.