SCHEMBL4190867

SCHEMBL4190867

NC(N)C(=O)c1cccc(O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.61
CA12 O43570 2/20 0.57
CA2 P00918 2/20 0.57
CA9 Q16790 2/20 0.57
CA1 P00915 1/20 0.57
CA6 P23280 1/20 0.57
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 2/20 0.55
EGLN2 Q96KS0 1/20 0.52
FASN P49327 1/20 0.48
CLK1 P49759 2/20 0.47
DYRK1A Q13627 2/20 0.47
DYRK1B Q9Y463 2/20 0.47
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
CA5A P35218 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CA5B Q9Y2D0 1/20 0.44
HSD17B1 P14061 6/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459041 0.84 PARP1 (0.57) PARP1CA12CA2CA9CA1
Hydrochloric Acid SCHEMBL6751733 0.82 PARP1 (0.55) PARP1CA12CA2CA9CA1
SCHEMBL28079434 0.79 GSK3B (0.58) PARP1CA12CA2CA9CA1
SCHEMBL21056000 0.79 CA12 (0.57) PARP1CA12CA2CA9CA1
SCHEMBL8084159 0.79 CA12 (0.57) PARP1CA12CA2CA9CA1
SCHEMBL3850377 0.78 CA12 (0.61) PARP1CA12CA2CA9CA1
Hydrochloric Acid SCHEMBL2569130 0.78 CA12 (0.55) PARP1CA12CA2CA9CA1
SCHEMBL28583896 0.78 CA12 (0.55) PARP1CA12CA2CA9CA1
SCHEMBL28007604 0.78 PARP1 (0.62) PARP1ALDH1A1GAAMAPTMEN1
SCHEMBL2989006 0.78 CA12 (0.55) PARP1CA12CA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130209515-A1 ANTI-INFECTIVE AND IMMUNOMODULATORY COMPOUNDS NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2013-08-15 US disclosed
US-20090215819-A1 ANTI-INFECTIVE AND IMMUNOMODULATORY COMPOUNDS NIH - DEITR 2009-08-27 US disclosed
WO-2006130832-A2 ANTI-INFECTIVE AND IMMUNOMODULATORY COMPOUNDS THE GENERAL HOSPITAL CORPORATION (US) 2006-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130209515-A1 ANTI-INFECTIVE AND IMMUNOMODULATORY COMPOUNDS IRF3, MAVS, MIF PARP1 2449/4885CA12 4135/4885CA2 4152/4885
US-20090215819-A1 ANTI-INFECTIVE AND IMMUNOMODULATORY COMPOUNDS IRF3, MAVS, MIF PARP1 2449/4885CA12 4135/4885CA2 4152/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.