SCHEMBL4191219

SCHEMBL4191219

COc1ccc2[nH]c3c(c2c1)CCCC3NCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.57
CDC42 P60953 1/20 0.54
GAA P10253 1/20 0.51
CASP6 P55212 1/20 0.51
CHRM4 P08173 1/20 0.51
DRD2 P14416 1/20 0.51
HTR7 P34969 1/20 0.51
PRMT5 O14744 2/20 0.50
CYP2D6 P10635 2/20 0.49
MAPT P10636 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HTR2B P41595 1/20 0.48
KCNH2 Q12809 1/20 0.48
ACHE P22303 1/20 0.47
MAPKAPK2 P49137 5/20 0.47
MAPKAPK5 Q8IW41 1/20 0.47
BRD3 Q15059 3/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4161906 0.99 SIRT1 (0.56) SIRT1CDC42GAACASP6CHRM4
SCHEMBL21998616 0.88 PRMT5 (0.54) SIRT1CDC42GAACASP6PRMT5
SCHEMBL4196258 0.87 RB1 (0.54) CDC42GAACASP6CHRM4DRD2
SCHEMBL5428515 0.86 GAA (0.64) SIRT1CDC42GAACASP6PRMT5
Hydrochloric Acid SCHEMBL4153475 0.86 RB1 (0.55) CDC42GAACASP6CHRM4DRD2
SCHEMBL5456604 0.86 GAA (0.69) SIRT1CDC42GAACASP6PRMT5
SCHEMBL22135732 0.85 CYP2D6 (0.55) SIRT1CDC42GAACASP6PRMT5
SCHEMBL22135730 0.85 CYP2D6 (0.55) SIRT1CDC42GAACASP6PRMT5
SCHEMBL22135752 0.85 CYP2D6 (0.55) SIRT1CDC42GAACASP6CHRM4
SCHEMBL22135751 0.85 CYP2D6 (0.55) SIRT1CDC42GAACASP6CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658068-B1 NOVEL CYCLOALKYL[B] CONDENSED INDOLES SMITHKLINE BEECHAM CORP (US) 2009-02-18 EP claimed
US-7622494-B2 Chemical compounds SMITHKLINE BEECHAM CORPORATION (US) 2009-11-24 US disclosed
US-7622494-B2 Chemical compounds SMITHKLINE BEECHAM CORPORATION (US) 2009-11-24 US disclosed
US-20090170923-A1 HCV INHIBITORS SMITHKLINE BEECHAM CORPORATION 2009-07-02 US disclosed
US-20090170923-A1 HCV INHIBITORS SMITHKLINE BEECHAM CORPORATION 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170923-A1 HCV INHIBITORS HAVCR2, MAVS, EIF2AK2 SIRT1 418/4885CDC42 1350/4885GAA 908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.