SCHEMBL4194616

SCHEMBL4194616

CC(C)Oc1ccc(I)cc1C(=O)NC(CC#N)Cc1c[nH]c2ccccc12.CC(C)Oc1ccc(I)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.45
ITGB2 P05107 6/20 0.43
ICAM1 P05362 6/20 0.43
ITGAL P20701 6/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
CTSC P53634 1/20 0.42
MAPT P10636 3/20 0.41
KDM4E B2RXH2 3/20 0.41
POLB P06746 2/20 0.41
APAF1 O14727 1/20 0.41
RECQL P46063 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
ECE1 P42892 3/20 0.40
ACE P12821 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944251 0.97 CTSL (0.45) CTSLITGB2ICAM1ITGALMEN1
SCHEMBL4169038 0.90 ITGB2 (0.45) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL3939262 0.86 MEN1 (0.46) ITGB2ICAM1ITGALMEN1KMT2A
SCHEMBL3937917 0.86 ITGB2 (0.46) CTSLITGB2ICAM1ITGALMEN1
SCHEMBL4041042 0.84 CTSL (0.42) CTSLITGB2ICAM1ITGALCTSS
SCHEMBL13905416 0.84 KMT2A (0.52) CTSLITGB2ICAM1ITGALMEN1
SCHEMBL3941203 0.83 ITGB2 (0.48) CTSLITGB2ICAM1ITGALMEN1
SCHEMBL13914323 0.82 CTSL (0.46) CTSLMEN1KMT2ACTSSCTSK
SCHEMBL13914332 0.82 HPGDS (0.47) CTSLITGB2ICAM1ITGALMEN1
SCHEMBL4041218 0.81 CTSL (0.44) CTSLMEN1KMT2ACTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016253-A2 CYANOMETHYL SUBSTITUTED N-ACYL TRYPTAMINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-02-05 WO disclosed