SCHEMBL4196829

SCHEMBL4196829

Cc1ccc(C(=O)N2CCC(c3ccc(C(F)(F)F)cc3)CC2)cc1N(CCNC(=O)OC(C)(C)C)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 3/20 0.45
EGLN1 Q9GZT9 1/20 0.41
GAA P10253 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
FASN P49327 5/20 0.40
CNR2 P34972 1/20 0.39
LMNA P02545 1/20 0.39
NPC1L1 Q9UHC9 3/20 0.39
SLC9A1 P19634 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRB3 P13945 1/20 0.38
HRH2 P25021 1/20 0.38
SLC6A4 P31645 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR2B P41595 1/20 0.38
HTR6 P50406 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
PROKR1 Q8TCW9 2/20 0.38
CNR1 P21554 1/20 0.38
CHRM2 P08172 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4202422 0.88 FASN (0.50) FASN
SCHEMBL4203527 0.84 FASN (0.49) FASN
SCHEMBL4204882 0.83 FASN (0.48) FASN
SCHEMBL4738015 0.81 PARP10 (0.46) EGLN1FASNLMNA
SCHEMBL4196832 0.81 P2RY14 (0.47) P2RY14EGLN1FASNCNR2NPC1L1
SCHEMBL4738617 0.79 PARP10 (0.45) FASNLMNASLC9A1PROKR1
SCHEMBL4201395 0.78 FASN (0.50) FASN
SCHEMBL4203212 0.77 FASN (0.53) FASN
SCHEMBL4207436 0.76 FASN (0.52) FASN
SCHEMBL4739507 0.76 FASN (0.52) FASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090118332-A1 Therapeutic Agents - 551 ASTRAZENECA AB (SE) 2009-05-07 US disclosed
WO-2008075064-A1 PIPERIDINE DERIVATIVES FOR THE TREATMENT OF OBESITY ASTRAZENECA AB (SE) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118332-A1 Therapeutic Agents - 551 GPR119, FABP4, FASN P2RY14 3232/4885EGLN1 551/4885GAA 393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.