SCHEMBL4199218

SCHEMBL4199218

CC(=O)N(C)CCN(C(N)=O)c1cc(C(=O)N2CCC(c3ccc(F)cc3)CC2)ccc1C

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 4/20 0.47
PARP14 Q460N5 2/20 0.47
ALDH1A1 P00352 2/20 0.41
FASN P49327 5/20 0.41
NAMPT P43490 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.40
HTR7 P34969 1/20 0.40
PROKR1 Q8TCW9 1/20 0.40
HSD11B1 P28845 2/20 0.39
LSS P48449 1/20 0.39
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4207291 0.89 FASN (0.53) FASN
SCHEMBL4738617 0.88 PARP10 (0.45) PARP10PARP14ALDH1A1FASNNAMPT
SCHEMBL4738015 0.87 PARP10 (0.46) PARP10PARP14ALDH1A1FASNNAMPT
SCHEMBL4193256 0.80 FASN (0.51) FASN
SCHEMBL4199222 0.77 FASN (0.45) PARP10FASN
SCHEMBL4199414 0.77 FASN (0.54) FASN
SCHEMBL4202879 0.76 FASN (0.55) FASN
SCHEMBL4199547 0.76 FASN (0.53) FASN
SCHEMBL4191753 0.75 PARP10 (0.58) PARP10PARP14ALDH1A1FASNNAMPT
SCHEMBL4204850 0.75 PARP14 (0.42) PARP10PARP14ALDH1A1FASNHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090118332-A1 Therapeutic Agents - 551 ASTRAZENECA AB (SE) 2009-05-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118332-A1 Therapeutic Agents - 551 GPR119, FABP4, FASN PARP10 1851/4885PARP14 1838/4885ALDH1A1 321/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.