SCHEMBL20103340

SCHEMBL20103340

CON(C)C(=O)c1cncc(OCc2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
HTT P42858 1/20 0.49
GFER P55789 1/20 0.49
HSD17B10 Q99714 1/20 0.49
SIRT2 Q8IXJ6 13/20 0.48
SIRT3 Q9NTG7 10/20 0.48
SIRT1 Q96EB6 8/20 0.48
MAOB P27338 2/20 0.48
NR4A2 P43354 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30678236 0.83 MAOB (0.66) KMT2AMEN1MAOBNR4A2
SCHEMBL4200015 0.83 MAOB (0.66) KMT2AMEN1MAOBNR4A2
SCHEMBL1202881 0.82 SIRT2 (0.59) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL7413175 0.81 CYP11B1 (0.42) KMT2AHTTSIRT2SIRT3SIRT1
SCHEMBL1034311 0.81 MAOB (0.63) KMT2AMEN1MAOBNR4A2
SCHEMBL1201866 0.81 MEN1 (0.70) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL30822583 0.81 MEN1 (0.70) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL2197204 0.80 MEN1 (0.68) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL3358456 0.80 APP (0.60) SIRT2SIRT3SIRT1MAOB
SCHEMBL3358460 0.80 APP (0.60) SIRT2SIRT3SIRT1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10988433-B2 Cyclohexyl GPR40 agonists for the treatment of type II diabetes JANSSEN PHARMACEUTICA NV (BE) 2021-04-27 US disclosed
US-20200039914-A1 CYCLOHEXYL GPR40 AGONISTS FOR THE TREATMENT OF TYPE II DIABETES JANSSEN RESEARCH & DEVELOPMENT, LLC 2020-02-06 US disclosed
WO-2018081047-A1 CYCLOHEXYL GPR40 AGONISTS FOR THE TREATMENT OF TYPE II DIABETES JANSSEN PHARMACEUTICA NV (BE) 2018-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200039914-A1 CYCLOHEXYL GPR40 AGONISTS FOR THE TREATMENT OF TYPE II DIABETES GPR119, GPR65, GPR55 KMT2A 3114/4885MEN1 4514/4885HTT 3053/4885
US-10988433-B2 Cyclohexyl GPR40 agonists for the treatment of type II diabetes GPR119, GPR65, GPR55 KMT2A 3114/4885MEN1 4514/4885HTT 3053/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.