SCHEMBL4200757

SCHEMBL4200757

O=NNCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.47
ALDH1A1 P00352 1/20 0.46
MTOR P42345 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
LSS P48449 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
IDO1 P14902 2/20 0.42
ASPH Q12797 1/20 0.42
KDM8 Q8N371 1/20 0.42
PPARA Q07869 1/20 0.41
MAPK14 Q16539 1/20 0.41
EPHX2 P34913 1/20 0.41
KIF11 P52732 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6232801 0.79 FFAR1 (0.44) FFAR1ALDH1A1MTORTAAR1HDAC3
SCHEMBL1436108 0.76 PTPN1 (0.54) FFAR1ALDH1A1MTORTAAR1IDO1
SCHEMBL3310761 0.76 ADH1B (0.55) FFAR1ALDH1A1MTORTAAR1HDAC3
SCHEMBL7345712 0.75 FFAR1 (0.68) FFAR1ALDH1A1MTORPPARA
SCHEMBL25588013 0.74 ALDH1A1 (0.52) FFAR1ALDH1A1MTORTAAR1HDAC3
SCHEMBL27982876 0.74 ALDH1A1 (0.52) FFAR1ALDH1A1MTORTAAR1HDAC3
Hydrochloric Acid SCHEMBL7347655 0.74 IDO1 (0.52) FFAR1ALDH1A1MTORTAAR1HDAC3
SCHEMBL29026424 0.73 FFAR1 (0.49) FFAR1MTORHDAC3HDAC1HDAC2
SCHEMBL296280 0.72 ALDH1A1 (0.55) ALDH1A1TAAR1LSSIDO1KIF11
SCHEMBL20058285 0.72 TAAR1 (0.48) ALDH1A1TAAR1HDAC1HDAC8IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828223-A4 NOVEL BETULIN DERIVATIVES, PREPARATION THEREOF AND USE THEREOF PANACOS PHARMACEUTICALS INC (US) 2009-03-11 EP disclosed
EP-1828223-A2 NOVEL BETULIN DERIVATIVES, PREPARATION THEREOF AND USE THEREOF Panacos Pharmaceuticals, Inc. (US) 2007-09-05 EP disclosed
WO-2006053255-A2 NOVEL BETULIN DERIVATIVES, PREPARATION THEREOF AND USE THEREOF PANACOS PHARMACEUTICALS, INC. (US) 2006-05-18 WO disclosed