SCHEMBL4200799

SCHEMBL4200799

O=Cc1cnnn1Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.48
P2RX7 Q99572 1/20 0.47
IDO1 P14902 2/20 0.42
CDC7 O00311 1/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
SLC9A1 P19634 1/20 0.41
GRM2 Q14416 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RECQL P46063 1/20 0.41
KDM4E B2RXH2 2/20 0.40
HPGD P15428 1/20 0.40
CYP19A1 P11511 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
TSHR P16473 1/20 0.39
TDO2 P48775 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15875591 0.77 HSD11B1 (0.51) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL1646429 0.75 P2RX7 (0.60) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL2895624 0.75 CDC7 (0.54) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL27676262 0.74 P2RX7 (0.46) P2RX7IDO1ALDH1A1LMNASLC9A1
SCHEMBL28230792 0.73 P2RX7 (0.50) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL11563985 0.73 P2RX7 (0.50) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL1371186 0.73 KDM4E (0.54) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL23336762 0.72 HSD11B1 (0.55) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL2895467 0.71 CDC7 (0.61) HSD11B1P2RX7IDO1CDC7ALDH1A1
SCHEMBL4195851 0.71 HSD11B1 (0.61) HSD11B1P2RX7IDO1CDC7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095394-A1 DIAZEPANES AS HISTAMINE H3 RECEPTOR ANTAGONISTS EVOTEC NEUROSCIENCES GMBH (DE) 2009-08-06 WO disclosed
WO-2009095394-A1 DIAZEPANES AS HISTAMINE H3 RECEPTOR ANTAGONISTS EVOTEC NEUROSCIENCES GMBH (DE) 2009-08-06 WO disclosed