SCHEMBL4203753

SCHEMBL4203753

NC1CNc2ccccc2[N]C1=O

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4203755 1.00 ALDH1A1 (0.31) ALDH1A1LMNAMAPT
SCHEMBL12345838 0.69 CREBBP (0.44) ALDH1A1MAPT
SCHEMBL6308518 0.69 CREBBP (0.44) ALDH1A1MAPT
SCHEMBL38765 0.68 BRPF1 (0.39) ALDH1A1LMNAMAPT
Hydrochloric Acid SCHEMBL2235061 0.68 CREBBP (0.43) ALDH1A1MAPT
Hydrochloric Acid SCHEMBL2235068 0.68 CREBBP (0.43) ALDH1A1MAPT
SCHEMBL129351 0.67 HTR2A (0.37)
SCHEMBL1592807 0.66 MEN1 (0.40) ALDH1A1LMNAMAPT
SCHEMBL8904356 0.66 GAA (0.39) ALDH1A1MAPT
SCHEMBL3913695 0.64 KDM1A (0.38) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083014-A2 Inhibitors of interleukin-1ß converting enzyme Vertex Pharmceuticals Incorporated (US) 2009-07-29 EP disclosed