SCHEMBL4210095

SCHEMBL4210095

BrCCCn1cc2ccccc2c1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.33
CCND1 P24385 4/20 0.33
TDP1 Q9NUW8 1/20 0.31
CYP2A6 P11509 1/20 0.30
ALOX12 P18054 1/20 0.30
SOD1 P00441 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30179235 0.93 CDK4 (0.36) CDK4CCND1TDP1
SCHEMBL6426597 0.91 CDK4 (0.38) CDK4CCND1
SCHEMBL3632871 0.86 BCHE (0.34) CDK4CCND1TDP1CYP2A6ALOX12
SCHEMBL11801475 0.77 HEXA (0.42)
SCHEMBL29351222 0.75 CYP2A6 (0.37) CDK4CCND1TDP1CYP2A6ALOX12
SCHEMBL9385329 0.74 CDK4 (0.38) CDK4CCND1
SCHEMBL377726 0.71 CDK4 (0.33) CDK4CCND1CYP2A6ALOX12
SCHEMBL7004471 0.71 HTR2A (0.38) CDK4CCND1CYP2A6ALOX12
SCHEMBL608395 0.71 LMNA (0.49)
SCHEMBL7365093 0.71 FABP4 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103022-A1 DERIVATIVES OF SUBSTITUTED FUSED RING CYCLOINDOLES AND METHODS OF THEIR USE ITHERX PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed