SCHEMBL4225022

SCHEMBL4225022

O=C1NC(=O)c2cc(O)c(O)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.47
PRKD3 O94806 3/20 0.47
PRKCG P05129 3/20 0.47
PRKCB P05771 3/20 0.47
SRC P12931 3/20 0.47
PRKCA P17252 3/20 0.47
PRKCH P24723 3/20 0.47
PRKCI P41743 3/20 0.47
PRKCE Q02156 3/20 0.47
PRKCQ Q04759 3/20 0.47
PRKCZ Q05513 3/20 0.47
PRKCD Q05655 3/20 0.47
PRKD1 Q15139 3/20 0.47
ABL1 P00519 1/20 0.47
ABL2 P42684 1/20 0.47
PPOX P50336 1/20 0.46
GSK3B P49841 1/20 0.46
BCL2 P10415 2/20 0.44
MCL1 Q07820 2/20 0.44
BRAF P15056 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24414673 0.83 KDM4E (0.52) EGFRPRKD3PRKCGPRKCBSRC
SCHEMBL38656398 0.79 CA1 (0.44) EGFRPRKD3PRKCGPRKCBSRC
SCHEMBL8650681 0.75 HMGCR (0.46) PRKCIGSK3BTDP1MEN1MAPT
SCHEMBL30828317 0.74 MAOA (0.56) EGFRPRKD3PRKCGPRKCBSRC
SCHEMBL177986 0.74 MAOA (0.56) EGFRPRKD3PRKCGPRKCBSRC
SCHEMBL1081926 0.73 GRM5 (0.55) EGFRPRKD3PRKCGPRKCBSRC
SCHEMBL15638608 0.72 CES1 (0.57) EGFRBCL2MCL1TDP1MAPT
SCHEMBL15680364 0.71 PPOX (0.42) PPOXGSK3BBCL2MCL1PTGS2
SCHEMBL8821657 0.71 BCL2 (0.74) BCL2MCL1TDP1CYP3A4MEN1
SCHEMBL28805663 0.71 BCL2 (0.46) EGFRPRKD3PRKCGPRKCBSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026248-A2 HYDRAZIDE, AMIDE, PHTHALIMIDE AND PHTHALHYDRAZIDE ANALOGS AS INHIBITORS OF RETROVIRAL INTEGRASE THE GOVERNMENT OF THE UNITED STATES, AS REPRESENTED BY THE SECRETARY OF HEALTH AND HUMAN SERVICES, NATIONAL INSTITUTES OF HEALTH, OFFICE OF TECHNOLOGY TRANSFER (US) 2009-02-26 WO disclosed
EP-0412763-B1 Cephalosporins, processes for their preparation, pharmaceutical compositions containing them and intermediates therefor ZENECA LTD (GB) 1996-07-10 EP disclosed
US-5219848-A Bactericides ICI PHARMA (FR) 1993-06-15 US disclosed