SCHEMBL4233124

SCHEMBL4233124

c1ccc(COCCn2cc(-c3nsc(Nc4ccccn4)n3)cn2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
KDR P35968 5/20 0.35
GRM4 Q14833 2/20 0.33
P2RY1 P47900 1/20 0.33
KCNH2 Q12809 1/20 0.33
KAT6A Q92794 1/20 0.33
KAT5 Q92993 1/20 0.33
KAT8 Q9H7Z6 1/20 0.33
TP53 P04637 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MCL1 Q07820 1/20 0.32
SGMS2 Q8NHU3 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4239760 0.83 MET (0.38) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL4235797 0.81 KDR (0.40) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL4243041 0.77 SCD (0.43)
SCHEMBL4236523 0.77 EGFR (0.41) NPC1RAB9AMEN1KMT2ACASP3
Hydrochloric Acid SCHEMBL4234156 0.77 EGFR (0.41) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL4243830 0.76 EGFR (0.39) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL4241653 0.74 JAK2 (0.40) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL4241649 0.70 GRK2 (0.40) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL3359286 0.69 NPC1 (0.46) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL3354854 0.68 GRM4 (0.62) NPC1RAB9AMEN1KMT2ACASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO disclosed