SCHEMBL4243041

SCHEMBL4243041

Fc1cccc(Cn2cc(-c3nsc(Nc4ccccn4)n3)cn2)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCD O00767 5/20 0.43
ADORA2B P29275 13/20 0.43
ADORA3 P0DMS8 9/20 0.43
ADORA1 P30542 11/20 0.42
ADORA2A P29274 10/20 0.42
ALK Q9UM73 1/20 0.42
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
SCD5 Q86SK9 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4235797 0.81 KDR (0.40)
SCHEMBL4239760 0.79 MET (0.38)
SCHEMBL4233124 0.77 NPC1 (0.36)
SCHEMBL4236523 0.77 EGFR (0.41) ADORA2BADORA3ADORA1ADORA2A
Hydrochloric Acid SCHEMBL4234156 0.77 EGFR (0.41) ADORA2BADORA3ADORA1ADORA2A
SCHEMBL4243830 0.76 EGFR (0.39) ADORA3ADORA2ACDK5
SCHEMBL4241653 0.74 JAK2 (0.40) SCDCDK5
SCHEMBL4241649 0.70 GRK2 (0.40) ADORA3CDK5
SCHEMBL4239119 0.70 MEN1 (0.42) ADORA3CDK5CDK5R1
SCHEMBL3359286 0.69 NPC1 (0.46) ADORA3CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO claimed