SCHEMBL4241653

SCHEMBL4241653

c1ccc(Nc2nc(-c3cnn(CC4CCOCC4)c3)ns2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.40
JAK1 P23458 2/20 0.40
JAK3 P52333 2/20 0.40
TYK2 P29597 1/20 0.40
LRRK2 Q5S007 1/20 0.40
TTK P33981 1/20 0.38
EGFR P00533 1/20 0.37
MAP3K12 Q12852 1/20 0.37
IKBKE Q14164 1/20 0.36
TBK1 Q9UHD2 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
SCD O00767 1/20 0.35
FGFR1 P11362 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4236523 0.93 EGFR (0.41) TTKEGFRTBK1MEN1NPC1
Hydrochloric Acid SCHEMBL4234156 0.92 EGFR (0.41) TTKEGFRTBK1MEN1NPC1
SCHEMBL4243830 0.91 EGFR (0.39) LRRK2TTKEGFRTBK1MEN1
SCHEMBL4235797 0.81 KDR (0.40) JAK2MEN1NPC1CASP3RAB9A
SCHEMBL4239760 0.79 MET (0.38) MEN1NPC1CASP3RAB9AKMT2A
SCHEMBL4241553 0.76 CREBBP (0.43) TTKEGFRPIK3CDPIK3CAPIK3CB
SCHEMBL4241649 0.76 GRK2 (0.40) JAK2JAK1JAK3TYK2LRRK2
SCHEMBL4237571 0.74 EGFR (0.41) TTKEGFRFGFR1FGFR3FGFR2
SCHEMBL4233124 0.74 NPC1 (0.36) MEN1NPC1CASP3RAB9AKMT2A
SCHEMBL4243041 0.74 SCD (0.43) SCDCDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO disclosed