SCHEMBL4236945

SCHEMBL4236945

N#Cc1ccc2ccc(N(CC(=O)O)S(=O)(=O)c3cc(Cl)cc(Cl)c3)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 8/20 0.46
NFE2L2 Q16236 8/20 0.46
RORC P51449 2/20 0.43
DAGLA Q9Y4D2 1/20 0.41
HCRTR2 O43614 1/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
S1PR1 P21453 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 1/20 0.39
NR3C1 P04150 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237417 0.97 KEAP1 (0.46) KEAP1NFE2L2RORCDAGLAHCRTR2
SCHEMBL12115563 0.86 RORC (0.42) RORCHCRTR2NR3C1
SCHEMBL4239508 0.83 KEAP1 (0.44) KEAP1NFE2L2ALDH1A1L3MBTL1S1PR1
SCHEMBL12115526 0.82 RORC (0.42) RORCHCRTR2NR3C1
SCHEMBL1110128 0.79 KEAP1 (0.41) KEAP1NFE2L2RORCHCRTR2ALDH1A1
SCHEMBL3303970 0.78 CDC7 (0.39) KEAP1NFE2L2RORCDAGLAALDH1A1
SCHEMBL3303192 0.78 KEAP1 (0.37) KEAP1NFE2L2RORCDAGLAHCRTR2
SCHEMBL4240479 0.78 KEAP1 (0.39) KEAP1NFE2L2ALDH1A1L3MBTL1S1PR1
SCHEMBL1317802 0.77 KEAP1 (0.43) KEAP1NFE2L2RORCALDH1A1L3MBTL1
SCHEMBL1110188 0.77 PSEN1 (0.39) RORCHCRTR2ALDH1A1SMN1; SMN2NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009127723-A1 NEW ARYLSULPHONYLGLYCINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-22 WO disclosed