SCHEMBL4239508

SCHEMBL4239508

Nc1ccc2ccc(N(CC(=O)O)S(=O)(=O)c3cc(Cl)cc(Cl)c3)cc2c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 11/20 0.44
NFE2L2 Q16236 11/20 0.44
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
S1PR1 P21453 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12115554 0.85 PSEN1 (0.36) KEAP1NFE2L2S1PR1TP53
SCHEMBL4236945 0.83 KEAP1 (0.46) KEAP1NFE2L2ALDH1A1L3MBTL1S1PR1
SCHEMBL1317802 0.82 KEAP1 (0.43) KEAP1NFE2L2ALDH1A1L3MBTL1S1PR1
SCHEMBL13658664 0.81 PSEN1 (0.38) KEAP1NFE2L2S1PR1TP53
SCHEMBL4240479 0.80 KEAP1 (0.39) KEAP1NFE2L2ALDH1A1L3MBTL1S1PR1
SCHEMBL4237417 0.79 KEAP1 (0.46) KEAP1NFE2L2ALDH1A1L3MBTL1S1PR1
SCHEMBL3058248 0.79 S1PR1 (0.38) S1PR1
SCHEMBL4233539 0.79 NPC1 (0.47) KEAP1NFE2L2ALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL4236740 0.78 L3MBTL1 (0.47) KEAP1NFE2L2L3MBTL1
SCHEMBL1319761 0.78 KEAP1 (0.43) KEAP1NFE2L2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009127723-A1 NEW ARYLSULPHONYLGLYCINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-22 WO disclosed