SCHEMBL4239119

SCHEMBL4239119

COc1ccc(-n2cc(-c3nsc(Nc4ccccn4)n3)cn2)cc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CG P48736 1/20 0.38
JUN P05412 1/20 0.38
MAPK10 P53779 1/20 0.38
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
MAPT P10636 2/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4235797 0.72 KDR (0.40) MEN1KMT2ANPC1RAB9ACASP3
SCHEMBL4243041 0.70 SCD (0.43) ADORA3CDK5CDK5R1
SCHEMBL4239760 0.69 MET (0.38) MEN1KMT2ANPC1RAB9ACASP3
SCHEMBL3359286 0.69 NPC1 (0.46) MEN1KMT2ANPC1RAB9AMAPK10
SCHEMBL4241649 0.68 GRK2 (0.40) MEN1KMT2ANPC1RAB9ACASP3
SCHEMBL4243223 0.68 NPC1 (0.42) MEN1KMT2ANPC1RAB9AMAPK10
SCHEMBL4236523 0.68 EGFR (0.41) MEN1KMT2ANPC1RAB9APIK3CD
Hydrochloric Acid SCHEMBL4234156 0.67 EGFR (0.41) MEN1KMT2ANPC1RAB9APIK3CD
SCHEMBL12989108 0.67 ALDH1A1 (0.42) MEN1KMT2ARAB9AMAPTHTT
SCHEMBL3911186 0.67 ABCG2 (0.56) MEN1KMT2ANPC1RAB9APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO disclosed