SCHEMBL4240397

SCHEMBL4240397

N=C(N)NC(=O)CC1c2cc(CC(F)(F)F)ccc2C(=O)N1CC(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.33
KCNH2 Q12809 1/20 0.33
SCN5A Q14524 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4463902 0.87 P2RX7 (0.35) KCNH2
SCHEMBL4185595 0.87 ALDH1A1 (0.35) SCN9AKCNH2SCN5A
SCHEMBL1385654 0.87 ALDH1A1 (0.35) SCN9AKCNH2SCN5A
SCHEMBL4181329 0.87 ALDH1A1 (0.35) SCN9AKCNH2SCN5A
SCHEMBL4240395 0.84
SCHEMBL4466189 0.84 TOP1 (0.36) SCN9AKCNH2SCN5A
SCHEMBL4464870 0.83 RORC (0.31)
SCHEMBL4464877 0.83 RORC (0.31)
SCHEMBL4467263 0.83 RORC (0.31)
SCHEMBL4478396 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531569-B2 Process for preparing (3-oxo-2,3-dihydro-1H-isoindol-1-yl) acetylguanidine derivatives SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2009-05-12 US claimed