SCHEMBL4242253

SCHEMBL4242253

COc1nc(N2CCN(C(=O)O)CC2)n(-c2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.46
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 4/20 0.43
MEN1 O00255 2/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 2/20 0.40
GLA P06280 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SLC1A2 P43004 1/20 0.39
DCTPP1 Q9H773 1/20 0.39
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568463 0.86 GPR119 (0.50) ALDH1A1LMNAMAPTTP53POLB
SCHEMBL13117238 0.80 KHK (0.48) LMNAMAPT
SCHEMBL4242255 0.79 ALDH1A1 (0.42) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL3564931 0.71 CKS1B (0.54) ALDH1A1LMNAMAPTTP53
SCHEMBL631962 0.70 ALDH1A1 (0.69) ALDH1A1KMT2AMEN1LMNAMAPT
Hydrochloric Acid SCHEMBL5492248 0.69 ALDH1A1 (0.67) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL3560832 0.69 GPR119 (0.49) ALDH1A1LMNAMAPTTP53POLB
SCHEMBL13117125 0.69 GPR119 (0.49) ALDH1A1LMNAMAPTTP53
SCHEMBL4319359 0.68 KMT2A (0.63) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL3562191 0.68 GPR119 (0.48) ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010525-A2 DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS Brystol-Myers Squibb Company (US) 2009-01-07 EP disclosed
WO-2007127635-A2 DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-08 WO disclosed