SCHEMBL4242255

SCHEMBL4242255

CS(=O)(=O)c1nc(N2CCN(C(=O)O)CC2)n(-c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
USP2 O75604 3/20 0.40
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KMT2A Q03164 3/20 0.38
TSHR P16473 2/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38
MGLL Q99685 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562191 0.85 GPR119 (0.48) ALDH1A1TP53THRB
SCHEMBL13117233 0.82 HTR3E (0.45)
SCHEMBL4242253 0.79 ALDH1A1 (0.46) ALDH1A1USP2MAPTTP53LMNA
SCHEMBL631962 0.69 ALDH1A1 (0.69) ALDH1A1USP2MAPTLMNANPSR1
Hydrochloric Acid SCHEMBL5492248 0.68 ALDH1A1 (0.67) ALDH1A1USP2MAPTLMNANPSR1
SCHEMBL3564931 0.68 CKS1B (0.54) ALDH1A1MAPTTP53LMNATHRB
SCHEMBL27643066 0.66 AKR1C3 (0.68) MAPTKMT2AMEN1
SCHEMBL2890817 0.66 HTT (0.52) ALDH1A1USP2MAPTTP53LMNA
SCHEMBL13117125 0.65 GPR119 (0.49) ALDH1A1MAPTTP53LMNATHRB
SCHEMBL3560832 0.65 GPR119 (0.49) ALDH1A1MAPTTP53LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010525-B1 Diketo-piperazine and piperidine derivatives as antiviral agents BRISTOL MYERS SQUIBB CO (US) 2013-08-28 EP disclosed
EP-2010525-A2 DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS Brystol-Myers Squibb Company (US) 2009-01-07 EP disclosed
WO-2007127635-A2 DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-08 WO disclosed