SCHEMBL424831

SCHEMBL424831

Nc1n[nH]c2cc(Br)ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 10/20 1.00
JAK2 O60674 3/20 1.00
KDM4E B2RXH2 1/20 0.52
CYP3A4 P08684 1/20 0.52
GAA P10253 1/20 0.52
DYRK1A Q13627 4/20 0.52
ABL1 P00519 2/20 0.50
BCR P11274 2/20 0.50
AXL P30530 1/20 0.47
AURKA O14965 2/20 0.46
TGFBR1 P36897 2/20 0.46
ROCK1 Q13464 2/20 0.46
AURKB Q96GD4 2/20 0.46
CHUK O15111 1/20 0.46
RPS6KB1 P23443 1/20 0.46
CDK2 P24941 1/20 0.46
KDR P35968 1/20 0.46
SYK P43405 1/20 0.46
JAK3 P52333 1/20 0.46
MAP3K5 Q99683 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29549192 1.00 PDPK1 (1.00) PDPK1JAK2KDM4ECYP3A4GAA
SCHEMBL786329 0.83 JAK2 (1.00) PDPK1JAK2KDM4ECYP3A4GAA
Formic Acid Phenyl Ester SCHEMBL28129440 0.80 PDPK1 (0.63) PDPK1JAK2KDM4ECYP3A4GAA
SCHEMBL922069 0.78 PDPK1 (0.65) PDPK1JAK2KDM4ECYP3A4GAA
SCHEMBL31539770 0.78 PDPK1 (0.63) PDPK1JAK2DYRK1AAXLAURKB
SCHEMBL11034 0.78 PDPK1 (0.63) PDPK1JAK2DYRK1AAXLAURKB
SCHEMBL15288061 0.78 PDPK1 (0.63) PDPK1JAK2DYRK1AAXLAURKB
SCHEMBL15288471 0.78 PDPK1 (0.63) PDPK1JAK2DYRK1AAXLAURKB
SCHEMBL29490946 0.78 PDPK1 (0.63) PDPK1JAK2DYRK1AABL1AXL
SCHEMBL2302544 0.78 PDPK1 (0.63) PDPK1JAK2DYRK1AAXLAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 358 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122080001-A Perfluoroalkyl substituted pyrimido [1,2-b ] indazole ketone compound and preparation method thereof 2026-05-26 CN claimed
CN-114573567-B Indazole cyclotriazole compound and preparation method and application thereof 西安交通大学 2023-05-02 CN claimed
CN-114573567-A Indazole cyclic triazole compound and preparation method and application thereof 西安交通大学 2022-06-03 CN claimed
CN-101962365-A Aminoindazole derivatives as protein-kinase inhibitors AVENTIS PHARMA SA 2011-02-02 CN claimed
CN-1656078-A Aminoindazole derivatives as protein kinase inhibitors AVENTIS PHARMA SA (FR) 2005-08-17 CN claimed
US-20040014802-A1 Aminoindazole derivatives and intermediates, preparation thereof, and pharmaceutical compositions thereof AVENTIS PHARMA S.A. (FR) 2004-01-22 US claimed
CN-122080001-A Perfluoroalkyl substituted pyrimido [1,2-b ] indazole ketone compound and preparation method thereof 2026-05-26 CN disclosed
EP-3870583-B1 SUBSTITUTED INDOLE AND INDAZOLE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2026-04-22 EP disclosed
US-12559492-B2 BRAF degraders C4 THERAPEUTICS, INC. (US) 2026-02-24 US disclosed
US-20260042782-A1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 THERAPEUTICS, INC. (US) 2026-02-12 US disclosed
US-20260021095-A1 BIFUNCTIONAL COMPOUNDS CONTAINING PYRIDO[2,3-d]PYRIMIDIN-7(8H)-ONE DERIVATIVES FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEASOME PATHWAY NIKANG THERAPEUTICS INC (US) 2026-01-22 US disclosed
EP-4681715-A2 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 Therapeutics, Inc. (US) 2026-01-21 EP disclosed
EP-4076450-B1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR C4 THERAPEUTICS INC (US) 2025-12-10 EP disclosed
US-6610677-B2 Enhancing glycogen synthesis, lowering blood levels of glucose, treating colon, ovarian, or breast cancer, treating diabetes, treating schizophrenia VERTEX PHARMACEUTICALS INCORPORATED 2003-08-26 US disclosed
US-20030083327-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2003-05-01 US disclosed
US-20030078166-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2003-04-24 US disclosed
US-20030073687-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2003-04-17 US disclosed
US-20030064981-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2003-04-03 US disclosed
US-20030064982-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2003-04-03 US disclosed
US-20030055044-A1 Pyrazole compounds useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2003-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030064981-A1 Pyrazole compounds useful as protein kinase inhibitors AURKC, AURKA, GSK3A PDPK1 178/4885JAK2 456/4885KDM4E 975/4885
US-20040014802-A1 Aminoindazole derivatives and intermediates, preparation thereof, and pharmaceutical compositions thereof CYP2C8, NR0B2, NR2C2 PDPK1 4495/4885JAK2 1774/4885KDM4E 3563/4885
US-20260021095-A1 BIFUNCTIONAL COMPOUNDS CONTAINING PYRIDO[2,3-d]PYRIMIDIN-7(8H)-ONE DERIVATIVES FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEASOME PATHWAY PSMB2, PSMB7, MDM2 PDPK1 1180/4885JAK2 1686/4885KDM4E 1441/4885
US-12559492-B2 BRAF degraders BRAF, NRAS, HRAS PDPK1 2427/4885JAK2 1297/4885KDM4E 1258/4885
US-20030064982-A1 Pyrazole compounds useful as protein kinase inhibitors MAP3K20, CDK2, MAP2K2 PDPK1 139/4885JAK2 352/4885KDM4E 596/4885
US-20030083327-A1 Pyrazole compounds useful as protein kinase inhibitors AURKC, AURKA, GSK3B PDPK1 230/4885JAK2 690/4885KDM4E 921/4885
US-20030055044-A1 Pyrazole compounds useful as protein kinase inhibitors AURKC, AURKA, GSK3B PDPK1 159/4885JAK2 487/4885KDM4E 605/4885
US-20030073687-A1 Pyrazole compounds useful as protein kinase inhibitors AURKC, AURKA, GSK3B PDPK1 239/4885JAK2 464/4885KDM4E 1142/4885
US-20260042782-A1 ISOINDOLINONE AND INDAZOLE COMPOUNDS FOR THE DEGRADATION OF EGFR EGFR, ERBB2, ERBB3 PDPK1 3256/4885JAK2 640/4885KDM4E 2261/4885
US-20030078166-A1 Pyrazole compounds useful as protein kinase inhibitors GSK3B, GSK3A, GSKIP PDPK1 10/4885JAK2 553/4885KDM4E 1005/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.