SCHEMBL4249231

SCHEMBL4249231

O=C(O)c1ccc(C(=O)c2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 1.00
TDP1 Q9NUW8 2/20 0.88
MAPK1 P28482 2/20 0.70
POLB P06746 1/20 0.70
LMNA P02545 1/20 0.69
GAA P10253 1/20 0.69
L3MBTL1 Q9Y468 1/20 0.67
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
CES1 P23141 2/20 0.63
CA1 P00915 3/20 0.61
CA2 P00918 3/20 0.61
ALDH1A1 P00352 2/20 0.61
MAPT P10636 1/20 0.61
CES2 O00748 1/20 0.60
TSHR P16473 1/20 0.59
CA12 O43570 1/20 0.57
CA9 Q16790 1/20 0.57
CA14 Q9ULX7 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28148545 0.94 SRD5A2 (0.89) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL43476 0.94 TDP1 (1.00) SRD5A2TDP1MAPK1POLBLMNA
Terephthalic Acid SCHEMBL28023943 0.94 TDP1 (1.00) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL1566327 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL7553997 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL10439552 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL3860571 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL17332086 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL11331124 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA
4-Nitrobenzoic Acid SCHEMBL17332065 0.91 TDP1 (0.95) SRD5A2TDP1MAPK1POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294622-B A kind of isoandrographolide class compound and preparation method and application 华南理工大学 2017-06-06 CN disclosed
CN-105294622-A Isoandrographolide compound, preparing method thereof and application thereof UNIV SOUTH CHINA TECH 2016-02-03 CN disclosed
US-7491735-B2 Chemokine receptor binding compounds GENZYME CORPORATION (US) 2009-02-17 US disclosed
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
US-20050277670-A1 Chemokine receptor binding compounds ANORMED INC. 2005-12-15 US disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed
US-5464912-A Adduct with rodlike mesogenic moiety, adduct made by reacting polyepoxide with nitro/so/ compound having epoxy-reactive hydrogen; conversion of hydroxyl product to ether, ester, halide, urethane, ketone, alkane; reducing nitro/so/ to amine THE DOW CHEMICAL COMPANY (US) 1995-11-07 US disclosed
US-5412044-A Nitro group terminated mesogenic epoxy resin adducts THE DOW CHEMICAL COMPANY (US) 1995-05-02 US disclosed
US-5344898-A Curable composition with stilbene groups and molecular orientation THE DOW CHEMICAL COMPANY (US) 1994-09-06 US disclosed
US-5298575-A Consists of at least one compound having more than one vicinal epoxide group and at least one amine terminated adduct containing one or more mesogenic moities THE DOW CHEMICAL COMPANY (US) 1994-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277670-A1 Chemokine receptor binding compounds CCR5, CXCR3, CCL5 SRD5A2 2236/4885TDP1 4502/4885MAPK1 1005/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.