SCHEMBL4249247

SCHEMBL4249247

O=S(=O)(c1ccccc1)c1cc(-c2cccc3ccccc23)ccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.50
CA1 P00915 5/20 0.50
CA2 P00918 5/20 0.50
CA9 Q16790 5/20 0.50
MCL1 Q07820 2/20 0.48
FEN1 P39748 3/20 0.46
ALOX5AP P20292 1/20 0.46
ACMSD Q8TDX5 1/20 0.45
HTR6 P50406 2/20 0.42
EDNRB P24530 1/20 0.41
EDNRA P25101 1/20 0.41
ACLY P53396 1/20 0.41
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
PTGS2 P35354 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11161303 0.75 CA12 (0.72) CA12CA1CA2CA9MCL1
SCHEMBL11781981 0.74 CA12 (0.50) CA12CA1CA2CA9MCL1
SCHEMBL7265174 0.72 HTR6 (0.50) FEN1HTR6
SCHEMBL3249669 0.71 HTR6 (0.73) CA1CA2CA9FEN1HTR6
SCHEMBL6548757 0.69 ALDH1A1 (0.54) CA12CA1CA2HTR6
SCHEMBL6839467 0.69 CA12 (0.48) CA12CA1CA2CA9MCL1
SCHEMBL257771 0.68 MEN1 (0.46) CA12CA1CA2CA9MCL1
SCHEMBL15853165 0.68 CYP11B1 (0.52) CA12CA1CA2CA9MCL1
SCHEMBL29892474 0.68 ALDH1A1 (0.44) CA12CA1CA2CA9MCL1
SCHEMBL17847460 0.68 MCL1 (0.43) CA12CA1CA2CA9MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824817-B1 ARYLSULFONYLNAPHTHALENE DERIVATIVES AS 5HT2A ANTAGONISTS MERCK SHARP & DOHME (GB) 2009-02-04 EP disclosed