SCHEMBL4249670

SCHEMBL4249670

[AsH2]CCc1nc2ccccc2[nH]1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.75
NPC1 O15118 1/20 0.68
RAB9A P51151 1/20 0.68
DDAH1 O94760 1/20 0.63
CHRM1 P11229 1/20 0.62
PDE10A Q9Y233 2/20 0.60
GAA P10253 1/20 0.59
BCHE P06276 1/20 0.58
PKM P14618 1/20 0.56
HTT P42858 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL230157 0.90 POLB (0.84) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL7854448 0.86 POLB (0.92) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL7006523 0.86 POLB (1.00) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL30701864 0.84 POLB (0.96) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL7854826 0.84 POLB (0.96) POLBNPC1RAB9ADDAH1CHRM1
Hydrochloric Acid SCHEMBL8466213 0.84 DDAH1 (0.63) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL30701863 0.84 POLB (0.96) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL7856315 0.84 POLB (0.96) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL7856311 0.84 POLB (0.96) POLBNPC1RAB9ADDAH1CHRM1
SCHEMBL2331252 0.84 POLB (0.96) POLBNPC1RAB9ADDAH1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010535-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120098-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed