SCHEMBL4254046

SCHEMBL4254046

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OCC)C1c1ccc2c(c1)OCCO2

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
KDM4E B2RXH2 5/20 0.61
HPGD P15428 2/20 0.61
TSHR P16473 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
ABCC1 P33527 1/20 0.59
LMNA P02545 2/20 0.57
GAA P10253 2/20 0.57
HSD17B10 Q99714 1/20 0.57
ADORA3 P0DMS8 2/20 0.53
CACNA1F O60840 1/20 0.53
CACNA1D Q01668 1/20 0.53
CACNA1S Q13698 1/20 0.53
CACNA1C Q13936 1/20 0.53
MGAM O43451 1/20 0.52
AMY1A P0DUB6 1/20 0.52
SI P14410 1/20 0.52
MGAM2 Q2M2H8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14413639 0.84 ALDH1A1 (0.87) ALDH1A1TSHRSMN1; SMN2GAAHSD17B10
SCHEMBL9505147 0.83 ADRA2A (0.51) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL7817206 0.81 KDM4E (0.88) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL10617897 0.80 ADRA2A (0.59) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL5342395 0.79 ALDH1A1 (0.61) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL2999858 0.78 KDM4E (0.65) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL14413641 0.77 ALDH1A1 (1.00) ALDH1A1TSHRSMN1; SMN2LMNAGAA
SCHEMBL11379013 0.77 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL3032293 0.77 KDM4E (0.80) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2
SCHEMBL3038503 0.76 ABCC1 (0.72) ALDH1A1KDM4EHPGDTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9045428-B2 Substituted heterocyclic compounds GILEAD SCIENCES, INC. (US) 2015-06-02 US claimed
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed