SCHEMBL9505147

SCHEMBL9505147

COC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1ccc2c(c1)OCCO2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.51
ADRA2B P18089 2/20 0.51
ADRA2C P18825 2/20 0.51
ADRA1D P25100 2/20 0.51
ADRA1A P35348 2/20 0.51
ADRA1B P35368 2/20 0.51
TSHR P16473 3/20 0.50
PDE1C Q14123 2/20 0.50
ALDH1A1 P00352 3/20 0.49
HSD17B10 Q99714 3/20 0.49
KDM4E B2RXH2 3/20 0.49
HTT P42858 2/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ADORA3 P0DMS8 1/20 0.48
NOTCH1 P46531 1/20 0.48
HPGD P15428 2/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10617897 0.88 ADRA2A (0.59) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL4254046 0.83 ALDH1A1 (0.63) TSHRALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9505134 0.81 PDE1C (0.46) TSHRPDE1CALDH1A1HSD17B10KDM4E
SCHEMBL7265410 0.78 TSHR (0.65) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL28446552 0.78 ADRA2A (0.55) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7245308 0.77 NOTCH1 (0.41) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9504286 0.77 GAA (0.59) ADRA1ATSHRPDE1CALDH1A1HSD17B10
SCHEMBL6951320 0.76 ADORA3 (0.76) TSHRPDE1CALDH1A1HSD17B10KDM4E
SCHEMBL9401767 0.76 KDM4E (0.68) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9272854 0.76 CACNA1F (0.69) TSHRPDE1CALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed