SCHEMBL4254388

SCHEMBL4254388

Cc1ccc2c(c1)C1(NC(=O)NC1=O)C(=O)N2CCC(C)C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.41
SCN9A Q15858 1/20 0.37
ALDH1A1 P00352 6/20 0.35
MAPT P10636 4/20 0.35
POLB P06746 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 2/20 0.34
ALOX15 P16050 1/20 0.34
PKM P14618 1/20 0.33
CNR1 P21554 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4255794 0.88 AKR1B1 (0.46) AKR1B1ALDH1A1MAPTPOLBCNR1
SCHEMBL4259941 0.87 AKR1B1 (0.48) AKR1B1
SCHEMBL4260787 0.87 AKR1B1 (0.48) AKR1B1SCN9AALDH1A1MAPTLMNA
SCHEMBL4260190 0.84 AKR1B1 (0.52) AKR1B1SCN9AALDH1A1MAPTSMN1; SMN2
SCHEMBL4255427 0.83 MAPT (0.45) AKR1B1SCN9AALDH1A1MAPTSMN1; SMN2
SCHEMBL4164829 0.83 AKR1B1 (0.41) AKR1B1ALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL4167713 0.82 AKR1B1 (0.40) AKR1B1ALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL4170928 0.81 AKR1B1 (0.39) AKR1B1ALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL4169551 0.81 ALDH1A1 (0.51) AKR1B1ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL4171124 0.81 AKR1B1 (0.39) AKR1B1ALDH1A1MAPTPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090176851-A1 Use of Spiro [Imidazolidine-4, 3' -Indole] 2, 2', 5' (1H) Triones for Treatment of Conditions Associated with Vanilloid Receptor 1 ASTRAZENECA AB (SE) 2009-07-09 US claimed
US-20090176851-A1 Use of Spiro [Imidazolidine-4, 3' -Indole] 2, 2', 5' (1H) Triones for Treatment of Conditions Associated with Vanilloid Receptor 1 ASTRAZENECA AB (SE) 2009-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176851-A1 Use of Spiro [Imidazolidine-4, 3' -Indole] 2, 2', 5' (1H) Triones for Treatment of Conditions Associated with Vanilloid Receptor 1 TRPV1, TRPV2, TRPV3 AKR1B1 366/4885SCN9A 575/4885ALDH1A1 502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.