SCHEMBL4254890

SCHEMBL4254890

COc1cccc2c1CCN2Cc1c[nH]cn1.COc1cccc2c1N(Cc1c[nH]cn1)CC2.Cc1ccc2c(c1)CCN2Cc1c[nH]cn1.Cc1ccc2c(c1)N(Cc1c[nH]cn1)CC2.Clc1cccc2c1N(Cc1c[nH]cn1)CC2

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.35
TRPM5 Q9NZQ8 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
ALDH1A1 P00352 3/20 0.31
MEN1 O00255 2/20 0.31
GAA P10253 2/20 0.31
KMT2A Q03164 2/20 0.31
USP2 O75604 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TRPV1 Q8NER1 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4248456 0.83 ALDH1A1 (0.30) ALDH1A1SMN1; SMN2
SCHEMBL3822149 0.82 HTR6 (0.35) HTR6TRPM5HDAC1HDAC6ALDH1A1
SCHEMBL3526525 0.78 DRD2 (0.41)
SCHEMBL3524800 0.77 NOTUM (0.44) HTR6HDAC1HDAC6TRPV1
SCHEMBL3530367 0.75 NOTUM (0.40) TRPM5MTNR1AMTNR1BALDH1A1MEN1
SCHEMBL3526848 0.75 HDAC1 (0.40) TRPM5HDAC1HDAC6ALDH1A1MEN1
SCHEMBL3530642 0.75 NOTUM (0.39) TRPM5ALDH1A1MEN1KMT2AUSP2
SCHEMBL3524887 0.72 HDAC1 (0.49) HDAC1HDAC6
SCHEMBL3823511 0.71 FNTA (0.38) HTR6TRPM5HDAC1HDAC6MAPT
SCHEMBL3529275 0.71 NOTUM (0.39) HTR6TRPM5TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084152-A2 SUBSTITUTED 4-IMIDAZOLES F. Hoffmann-Roche AG (CH) 2009-08-05 EP claimed
WO-2008058867-A2 SUBSTITUTED 4-IMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2008-05-22 WO claimed