SCHEMBL4255744

SCHEMBL4255744

[CH2]CC(Cc1ccccc1)(Cc1cncs1)N(Cc1ccccc1)Cc1ccco1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.35
RECQL P46063 1/20 0.34
NPSR1 Q6W5P4 6/20 0.34
TSHR P16473 3/20 0.33
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
HTT P42858 2/20 0.33
LMNA P02545 2/20 0.33
USP2 O75604 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TP53 P04637 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TAS2R14 Q9NYV8 1/20 0.32
ADORA2A P29274 1/20 0.32
THRB P10828 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4255741 0.65 NPSR1 (0.37) MAPTRECQLNPSR1TSHRALDH1A1
SCHEMBL9389496 0.60 SLC6A3 (0.49) LMNA
SCHEMBL16523570 0.60 TSHR (0.51) MAPTNPSR1TSHRALDH1A1MEN1
SCHEMBL27825512 0.59 SLC6A3 (0.47)
SCHEMBL5790031 0.58 TSHR (0.52) MAPTNPSR1TSHRALDH1A1MEN1
SCHEMBL28141333 0.58 TSHR (0.54) TSHRLMNACYP3A4KDM4E
SCHEMBL11011825 0.57 MAPT (0.52) MAPTNPSR1TSHRALDH1A1MEN1
SCHEMBL7990268 0.57 TP53 (0.50) MAPTNPSR1ALDH1A1MEN1KMT2A
SCHEMBL8497082 0.56 MAPT (0.47) MAPTNPSR1TSHRALDH1A1MEN1
SCHEMBL7990266 0.55 ALDH1A1 (0.44) MAPTTSHRALDH1A1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP claimed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO claimed
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed