SCHEMBL4255872

SCHEMBL4255872

CCC(C)(c1cc2c(Cl)c(C)nn2c(=O)n1Cc1ccccc1)N(CCCN(C)C)C(=O)c1ccc(OC)cc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 1/20 0.38
ACHE P22303 1/20 0.38
OPRM1 P35372 1/20 0.37
ALDH1A1 P00352 1/20 0.36
KIF11 P52732 6/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
KLK1 P06870 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
TBXA2R P21731 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4245624 0.93 KIF11 (0.41) ALDH1A1KIF11
SCHEMBL4255912 0.93 KIF11 (0.40) ALDH1A1KIF11TDP1
SCHEMBL4252369 0.91 KIF11 (0.37) ACHEALDH1A1KIF11KMT2AMEN1
SCHEMBL4245137 0.91 KIF11 (0.45) ALDH1A1KIF11CHRM2CHRM3TDP1
SCHEMBL4255894 0.90 KIF11 (0.36) ALDH1A1KIF11
SCHEMBL4251311 0.88 KIF11 (0.36) ALDH1A1KIF11KMT2AMEN1
SCHEMBL4249153 0.88 KIF11 (0.40) KIF11TDP1
SCHEMBL4255871 0.80 KIF11 (0.43) PDE1BKIF11
SCHEMBL4255875 0.79 PTGDR2 (0.41) PDE1BACHEALDH1A1KIF11KMT2A
SCHEMBL4055444 0.77 KIF11 (0.39) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035426-A1 PYRAZOLOPYRIMIDONES 4SC AG (DE) 2009-03-18 EP disclosed
WO-2007144384-A1 PYRAZOLOPYRIMIDONES 4SC AG (DE) 2007-12-21 WO disclosed