SCHEMBL4255919

SCHEMBL4255919

COc1ccc(-c2csc(C3CCNCC3)n2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.44
JAK3 P52333 2/20 0.44
PTK2 Q05397 1/20 0.44
HPGDS O60760 1/20 0.44
CYP1B1 Q16678 4/20 0.42
CYP1A1 P04798 3/20 0.42
HTR2C P28335 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
JAK1 P23458 1/20 0.40
EIF4E P06730 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
BAZ2A Q9UIF9 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PLAT P00750 1/20 0.38
AMY1A P0DUB6 2/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL2973520 0.99 JAK2 (0.44) JAK2JAK3PTK2HPGDSCYP1B1
SCHEMBL4262081 0.87 CYP1A1 (0.59) HPGDSCYP1B1CYP1A1HTR2CMEN1
Bromide SCHEMBL2985795 0.86 CYP1A1 (0.57) HPGDSCYP1B1CYP1A1HTR2CMEN1
SCHEMBL2981407 0.82 NPC1 (0.41) CYP1B1CYP1A1MEN1KMT2ANPC1
SCHEMBL2979646 0.81 ALDH1A1 (0.42) CYP1B1CYP1A1NPC1RAB9AEIF4E
SCHEMBL4257174 0.80 RAB9A (0.60) HPGDSCYP1B1CYP1A1MEN1KMT2A
SCHEMBL5072503 0.80 ALDH1A1 (0.36) JAK2JAK3PTK2NPC1RAB9A
SCHEMBL27713695 0.80 HPGDS (0.45) JAK2JAK3PTK2HPGDSHTR2C
SCHEMBL2981957 0.80 ALDH1A1 (0.40) JAK2JAK3PTK2CYP1B1CYP1A1
Bromide SCHEMBL2972856 0.79 NPC1 (0.62) HPGDSCYP1B1CYP1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945635-B1 THIAZOLYL PIPERIDINE DERIVATIVES USEFUL AS H3 RECEPTOR MODULATORS HOFFMANN LA ROCHE (CH) 2009-05-06 EP disclosed