SCHEMBL4257958

SCHEMBL4257958

CCOC(=O)C1=C(C)Nc2[nH]ncc2C1c1ccccc1-c1cccc(C(C)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 6/20 0.46
KDM4E B2RXH2 4/20 0.43
HSD17B10 Q99714 3/20 0.43
ADORA3 P0DMS8 3/20 0.43
ALDH1A1 P00352 2/20 0.43
CASP1 P29466 1/20 0.43
CACNA1F O60840 3/20 0.43
CACNA1D Q01668 3/20 0.43
CACNA1S Q13698 3/20 0.43
CYP2C9 P11712 3/20 0.42
MEN1 O00255 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
KMT2A Q03164 2/20 0.42
HIF1A Q16665 2/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
GAA P10253 2/20 0.42
ABCB1 P08183 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3009358 0.79 CACNA1C (0.44) CACNA1CKDM4EHSD17B10ADORA3ALDH1A1
SCHEMBL3004149 0.76 ADORA3 (0.60) CACNA1CKDM4EHSD17B10ADORA3ALDH1A1
SCHEMBL2999733 0.74 KDM4E (0.45) CACNA1CKDM4EHSD17B10ADORA3ALDH1A1
SCHEMBL4265478 0.74 KDM4E (0.52) CACNA1CKDM4EHSD17B10ADORA3ALDH1A1
SCHEMBL2994478 0.73 CACNA1C (0.56) CACNA1CKDM4EHSD17B10ADORA3ALDH1A1
SCHEMBL3004313 0.72 ALDH1A1 (0.56) KDM4EHSD17B10ADORA3ALDH1A1CASP1
SCHEMBL3009592 0.71 KDM4E (0.46) KDM4EHSD17B10ADORA3ALDH1A1CASP1
SCHEMBL2993757 0.71 PDE1C (0.41) CACNA1CHSD17B10ADORA3ALDH1A1CYP3A4
SCHEMBL4059888 0.70 TSHR (0.54) HSD17B10ALDH1A1CYP2C9MEN1CYP1A2
SCHEMBL4252896 0.70 MAPT (0.48) CACNA1CKDM4EHSD17B10ADORA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed