SCHEMBL4258353

SCHEMBL4258353

COC(=O)C#Cc1cccc(C(=O)OC)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP3A4 P08684 2/20 0.49
MAPK1 P28482 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.47
TSHR P16473 1/20 0.47
CYP4F2 P78329 2/20 0.46
CYP4A11 Q02928 2/20 0.46
RAB9A P51151 4/20 0.45
POLB P06746 2/20 0.45
NPC1 O15118 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MKNK2 Q9HBH9 1/20 0.43
BLM P54132 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
XDH P47989 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14829396 0.87 ALDH1A1 (0.52) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL14829600 0.87 ALDH1A1 (0.45) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL10411912 0.85 ALDH1A1 (0.52) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL4672150 0.83 ALDH1A1 (0.51) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL1926585 0.83 TSHR (0.60) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL16720308 0.82 KDM4E (0.55) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL14829517 0.80 ALDH1A1 (0.40) ALDH1A1CYP3A4MAPK1LOXL2CYP4F2
SCHEMBL13545801 0.80 PTPN11 (0.55) ALDH1A1LOXL2TSHRRAB9ANPC1
SCHEMBL1800821 0.80 TSHR (0.53) ALDH1A1CYP3A4MAPK1LOXL2TSHR
SCHEMBL18569778 0.79 ALDH1A1 (0.48) ALDH1A1CYP3A4MAPK1LOXL2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8735630-B2 Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2014-05-27 US disclosed
US-20130178632-A1 Transition-Metal-Catalyzed Carbon-Nitrogen and Carbon-Carbon Bond-Forming Reactions MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2013-07-11 US disclosed
US-8378145-B2 Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2013-02-19 US disclosed
US-20090287016-A1 Transition-Metal-Catalyzed Carbon-Nitrogen and Carbon-Carbon Bond-Forming Reactions MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2009-11-19 US disclosed
US-7560596-B2 Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2009-07-14 US disclosed
EP-1833605-A2 TRANSITION-METAL-CATALYZED CARBON-NITROGEN AND CARBON-CARBON BOND-FORMING REACTIONS Massachusetts Institute of Technology (US) 2007-09-19 EP disclosed
US-20060173186-A1 Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2006-08-03 US disclosed
WO-2006074315-A2 TRANSITION-METAL-CATALYZED CARBON-NITROGEN AND CARBON-CARBON BOND-FORMING REACTIONS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2006-07-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090287016-A1 Transition-Metal-Catalyzed Carbon-Nitrogen and Carbon-Carbon Bond-Forming Reactions NBAS, APEX1, CBR3 ALDH1A1 1530/4885CYP3A4 704/4885MAPK1 2488/4885
US-20060173186-A1 Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions NBAS, APEX1, CBR3 ALDH1A1 1530/4885CYP3A4 704/4885MAPK1 2488/4885
US-20130178632-A1 Transition-Metal-Catalyzed Carbon-Nitrogen and Carbon-Carbon Bond-Forming Reactions NBAS, APEX1, CBR3 ALDH1A1 1530/4885CYP3A4 704/4885MAPK1 2488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.