SCHEMBL4261

SCHEMBL4261

CC(C)(C)CNC(=O)N(CCl)N=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
BLM P54132 2/20 0.44
PMP22 Q01453 2/20 0.44
MEN1 O00255 1/20 0.44
ABCB11 O95342 1/20 0.44
GSR P00390 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
ADRA2A P08913 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE4A P27815 1/20 0.33
ADRA1A P35348 1/20 0.33
LMNA P02545 1/20 0.32
NFKB1 P19838 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentamustine SCHEMBL11151237 0.86 ALDH1A1 (0.64) ALDH1A1BLMPMP22MEN1ABCB11
SCHEMBL11148768 0.79 ALDH1A1 (0.42) ALDH1A1BLMPMP22MEN1ABCB11
SCHEMBL13098674 0.69 CHRNB2 (0.42) ALDH1A1TSHR
SCHEMBL4866354 0.65 ALDH1A1 (0.48) ALDH1A1MEN1TSHRHTTKMT2A
SCHEMBL9013052 0.64 ALDH1A1 (0.57) ALDH1A1BLMPMP22MEN1ABCB11
SCHEMBL3677883 0.64
SCHEMBL27115231 0.63
SCHEMBL25763748 0.63 ALDH1A1 (0.58) ALDH1A1BLMPMP22MEN1ABCB11
SCHEMBL2824552 0.62 BCHE (0.36) SMN1; SMN2
SCHEMBL10005923 0.62 ALDH1A1 (0.77) ALDH1A1BLMPMP22MEN1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9800 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4524131-A1 SMALL MOLECULES FOR TREATING CANCER, INHABITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH AlonBio Ltd. (IL) 2025-03-19 EP claimed
US-12202803-B2 Small molecules for treating cancer, inhibiting chemokine activity and/or inducing cell death ALONBIO LTD. (IL) 2025-01-21 US claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
US-12109219-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2024-10-08 US claimed
WO-2024162488-A1 PHARMACEUTICAL COMPOSITION COMPRISING CUCURBITACIN D FOR PREVENTING OR TREATING NEUROPATHIC PAIN 주식회사 재인알앤피 2024-08-08 WO claimed
EP-4401780-A1 AMORPHOUS PHOTOSENSITIZING PARTICLES, METHODS FOR THE PREPARATION THEREOF, AND METHODS FOR THE USE THEREOF University of Maryland, College Park (US) 2024-07-24 EP claimed
WO-2024026505-A2 DISRUPTION OF TELOCYTE ACTIVITY PATEL AMIT (US) 2024-02-01 WO claimed
US-20240002347-A1 SMALL MOLECULES FOR TREATING CANCER, INHIBITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH ALONBIO LTD. (IL) 2024-01-04 US claimed
CN-1628852-A Anti solid tumor medicine composition KONG QINGZHONG (CN) 2005-06-22 CN claimed
CN-1628849-A Anticancer medicine composition KONG QINGZHONG (CN) 2005-06-22 CN claimed
CN-1616098-A Anti-cancer medicine composition KONG QINGZHONG (CN) 2005-05-18 CN claimed
CN-1616099-A Anti-cancer medicine composition KONG QINGZHONG (CN) 2005-05-18 CN claimed
US-20040092583-A1 Treatment for inhibiting neoplastic lesions SHANAHAN-PRENDERGAST ELIZABETH (IE) 2004-05-13 US claimed
EP-1351678-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS Shanahan-Prendergast, Elizabeth (IE) 2003-10-15 EP claimed
US-20030072794-A1 Encapsulation of plasmid DNA (lipogenes™) and therapeutic agents with nuclear localization signal/fusogenic peptide conjugates into targeted liposome complexes REGULON, INC. 2003-04-17 US claimed
EP-1292284-A2 ENCAPSULATION OF POLYNUCLEOTIDES AND DRUGS INTO TARGETED LIPOSOMES Boulikas, Teni (US) 2003-03-19 EP claimed
WO-2002053138-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS SHANAHAN-PRENDERGAST ELISABETH (IE) 2002-07-11 WO claimed
WO-2001093836-A2 ENCAPSULATION OF POLYNUCLEOTIDES AND DRUGS INTO TARGETED LIPOSOMES BOULIKAS TENI (US) 2001-12-13 WO claimed