SCHEMBL4262107

SCHEMBL4262107

Cc1cccc(-c2cc(F)c3c(c2)NC(=O)CO3)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 9/20 0.51
PGR P06401 9/20 0.51
NR3C1 P04150 5/20 0.51
MMP12 P39900 1/20 0.46
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
PKM P14618 2/20 0.41
MAPK1 P28482 1/20 0.41
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRB2 P07550 2/20 0.40
ADRB1 P08588 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4263576 0.87 NR3C2 (0.50) NR3C2PGRNR3C1MMP12PDE3B
SCHEMBL4261432 0.86 NR3C2 (0.49) NR3C2PGRNR3C1MMP12PDE3B
SCHEMBL4265400 0.85 NR3C2 (0.53) NR3C2PGRNR3C1HTR1AHTR1D
SCHEMBL18305164 0.83 PGR (0.47) NR3C2PGRNR3C1PKMMAPK1
SCHEMBL13932102 0.79 MAOB (0.48) NR3C2PGRNR3C1MMP12PKM
SCHEMBL4267840 0.79 MAOB (0.48) NR3C2PGRNR3C1MMP12PKM
SCHEMBL12116980 0.79 PDE3B (0.53) NR3C2PGRNR3C1MMP12PDE3B
SCHEMBL4267366 0.79 MMP12 (0.70) NR3C2PGRNR3C1MMP12PDE3B
SCHEMBL18305051 0.79 CYP11B1 (0.60) NR3C2PGRNR3C1PDE3BPDE3A
SCHEMBL4272395 0.77 PGR (0.49) NR3C2PGRNR3C1MMP12HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090054417-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF STEROID HORMONE NUCLEAR RECEPTORS IRM LLC (BM) 2009-02-26 US claimed
US-20090054417-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF STEROID HORMONE NUCLEAR RECEPTORS IRM LLC (BM) 2009-02-26 US disclosed
US-20090054417-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF STEROID HORMONE NUCLEAR RECEPTORS IRM LLC (BM) 2009-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054417-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF STEROID HORMONE NUCLEAR RECEPTORS NR5A1, ESRRA, NR3C1 NR3C2 7/4885PGR 46/4885NR3C1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.