SCHEMBL4263337

SCHEMBL4263337

O=C(O)OC1=CS[C@@H]2/C(=C\c3cn4c(n3)sc3cc(F)ccc34)C(=O)N12

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.36
TP53 P04637 2/20 0.36
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4262075 0.90 PARP15 (0.36) MAPTTP53THRB
SCHEMBL4267704 0.86
SCHEMBL4263334 0.86
SCHEMBL4267705 0.79
SCHEMBL4259772 0.79 BRPF1 (0.36)
SCHEMBL4257558 0.76
SCHEMBL4257282 0.76 PARP15 (0.38)
SCHEMBL4254592 0.76 PARP15 (0.38) MAPT
SCHEMBL4261702 0.76 NPC1 (0.37) MAPTTP53
SCHEMBL4259319 0.76 NPC1 (0.35) MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499622-B1 HETEROTRICYCLYL 6-ALKYLIDENE-PENEMS AS BETA-LACTAMASE INHIBITORS WYETH CORP (US) 2009-03-11 EP claimed