SCHEMBL4268486

SCHEMBL4268486

Cc1ccccc1NC(=O)C=CC1=C(Cl)c2ccccc2CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 5/20 0.53
MMP2 P08253 5/20 0.53
MMP9 P14780 5/20 0.53
EGFR P00533 2/20 0.53
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
MAPT P10636 3/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
XBP1 P17861 1/20 0.43
KMT2A Q03164 1/20 0.43
TLR9 Q9NR96 1/20 0.43
ESR1 P03372 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4268646 0.85 MMP1 (0.56) MMP1MMP2MMP9EGFRNPC1
SCHEMBL4412018 0.83 MMP1 (0.53) MMP1MMP2MMP9EGFRNPC1
SCHEMBL4418306 0.79 MMP1 (0.53) MMP1MMP2MMP9EGFRNPC1
SCHEMBL4263459 0.78 MMP1 (0.56) MMP1MMP2MMP9EGFRNPC1
SCHEMBL4264174 0.76 ESR1 (0.50) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL4551139 0.76 ESR1 (0.50) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL4267886 0.76 ALDH1A1 (0.47) SMN1; SMN2MAPTKDM4EMEN1KMT2A
SCHEMBL4552432 0.76 MAPT (0.43) MMP1MMP2MMP9EGFRNPC1
SCHEMBL4429251 0.75 EGFR (0.49) EGFRMAPTLMNAKMT2AESR1
SCHEMBL4410001 0.75 MMP1 (0.53) MMP1MMP2MMP9NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO claimed
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO disclosed