SCHEMBL4552432

SCHEMBL4552432

O=C(O)C=CC1=C(Cl)c2ccccc2CC1.O=C(O)Nc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
ESR1 P03372 2/20 0.42
GAA P10253 1/20 0.41
RAB9A P51151 4/20 0.40
MITF O75030 1/20 0.40
HSP90AA1 P07900 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PKM P14618 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
NPC1 O15118 3/20 0.37
MAOB P27338 2/20 0.37
MAPK14 Q16539 2/20 0.37
KMT2A Q03164 1/20 0.36
EGFR P00533 2/20 0.35
MMP1 P03956 2/20 0.35
MMP2 P08253 2/20 0.35
MMP9 P14780 2/20 0.35
MAOA P21397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenylamine SCHEMBL4414722 0.90 ESR1 (0.44) MAPTESR1GAARAB9AMITF
SCHEMBL4264174 0.89 ESR1 (0.50) MAPTESR1GAARAB9AMITF
SCHEMBL4551139 0.89 ESR1 (0.50) MAPTESR1GAARAB9AMITF
Diethylamine SCHEMBL4562983 0.82 MAPT (0.43) MAPTESR1GAARAB9AMITF
SCHEMBL4412018 0.81 MMP1 (0.53) MAPTRAB9ANPC1MAOBKMT2A
Methylpiperazine SCHEMBL4551702 0.78 MAPT (0.44) MAPTESR1GAARAB9AMITF
SCHEMBL4418306 0.78 MMP1 (0.53) MAPTESR1GAARAB9AL3MBTL1
SCHEMBL4277728 0.77 MEN1 (0.45) MAPTESR1GAARAB9AMITF
SCHEMBL4268486 0.76 MMP1 (0.53) MAPTESR1GAARAB9ANPC1
SCHEMBL4266901 0.76 RAB9A (0.48) MAPTRAB9AMITFHSP90AA1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO disclosed