SCHEMBL4269883

SCHEMBL4269883

O=CC(Br)Cc1cccnc1F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.36
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
MMP2 P08253 2/20 0.32
MMP9 P14780 2/20 0.32
MMP8 P22894 2/20 0.32
MMP13 P45452 2/20 0.32
KDM1A O60341 1/20 0.32
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
KDM4E B2RXH2 1/20 0.30
CYP1A2 P05177 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4764946 0.75 ALDH1A1 (0.41)
SCHEMBL13044957 0.73 GABRA1 (0.45) NAPRTMMP2MMP9MMP8MMP13
SCHEMBL1811013 0.73 NAPRT (0.41) NAPRTTRIM24TRIM33MMP2MMP9
SCHEMBL28705949 0.72
SCHEMBL6989753 0.70
SCHEMBL13925527 0.70
SCHEMBL844104 0.70
SCHEMBL7270961 0.69 CYP1A2 (0.54) NAPRTKDM4ECYP1A2MAPT
SCHEMBL31754264 0.69 CYP1A2 (0.54) NAPRTKDM4ECYP1A2MAPT
SCHEMBL5283008 0.69 CYP1A2 (0.54) NAPRTKDM4ECYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed