SCHEMBL4270709

SCHEMBL4270709

O=CN1CCC[C@@H]1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACE P12821 8/20 0.41
REN P00797 1/20 0.39
LMNA P02545 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555101 1.00 ACE (0.41) ACERENLMNACYP2C19HSD17B10
SCHEMBL698970 1.00 ACE (0.41) ACERENLMNACYP2C19HSD17B10
SCHEMBL23223889 0.94 MEN1 (0.38) ACE
SCHEMBL157964 0.94 MEN1 (0.38) ACE
SCHEMBL15904216 0.86
SCHEMBL16518728 0.85 ACE (0.53) ACERENLMNACYP2C19HSD17B10
SCHEMBL12658485 0.85 ACE (0.53) ACERENLMNACYP2C19HSD17B10
SCHEMBL12584754 0.81 CNR1 (0.34)
SCHEMBL14400492 0.81 CNR1 (0.34)
SCHEMBL8959051 0.81 AR (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130324555-A1 Method of use of pharmaceutical formulations for the treatment of apicomplexan diseases in animals WOOD RICHARD DELAREY (US) 2013-12-05 US claimed
US-20130150416-A1 Glutamate receptor modulators and therapeutic agents WOOD RICHARD D (US) 2013-06-13 US claimed
US-20090239919-A1 Glutamate receptor modulators and therapeutic agents WOOD RICHARD DELAREY 2009-09-24 US claimed
US-5770594-A ANTICHOLESTEROL AGENTS, INHIBITORS OF CHOLESTEROL SYNTHESIS PFIZER INC. (US) 1998-06-23 US claimed
WO-1996020184-A1 NAPHTHYL-BENZOXAZEPINES OR -BENZOTHIAZEPINES AS SQUALENE SYNTHETASE INHIBITORS PFIZER INC. (US) 1996-07-04 WO claimed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-111601798-A Bisamide sarcomere activating compound and use thereof 美国安进公司 2020-08-28 CN disclosed
US-8614205-B2 Glutamate receptor modulators and therapeutic agents WOOD RICHARD D (US) 2013-12-24 US disclosed
US-20130324555-A1 Method of use of pharmaceutical formulations for the treatment of apicomplexan diseases in animals WOOD RICHARD DELAREY (US) 2013-12-05 US disclosed
US-20130150416-A1 Glutamate receptor modulators and therapeutic agents WOOD RICHARD D (US) 2013-06-13 US disclosed
US-8211882-B2 Glutamate receptor modulators and therapeutic agents WOOD RICHARD DELAREY (US) 2012-07-03 US disclosed
WO-2011103524-A2 CYCLIC TETRAPEPTIDES AND THERAPEUTIC APPLICATIONS THEREOF PEPTADERM SP.Z.O.O. (PL) 2011-08-25 WO disclosed
US-7851439-B2 EFTU inhibitors or aminothiazoles and their uses NOVARTIS AG (CH) 2010-12-14 US disclosed
US-20090239919-A1 Glutamate receptor modulators and therapeutic agents WOOD RICHARD DELAREY 2009-09-24 US disclosed
US-20080221142-A1 useful in interfering with the life cycle of bacteria and in treating or preventing a bacterial infection NOVARTIS AG (CH) 2008-09-11 US disclosed
US-5770594-A ANTICHOLESTEROL AGENTS, INHIBITORS OF CHOLESTEROL SYNTHESIS PFIZER INC. (US) 1998-06-23 US disclosed
WO-1996020184-A1 NAPHTHYL-BENZOXAZEPINES OR -BENZOTHIAZEPINES AS SQUALENE SYNTHETASE INHIBITORS PFIZER INC. (US) 1996-07-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090239919-A1 Glutamate receptor modulators and therapeutic agents GRM5, GRM1, GRIK5 ACE 2281/4885REN 944/4885LMNA 4247/4885
US-20080221142-A1 useful in interfering with the life cycle of bacteria and in treating or preventing a bacterial infection LPO, PCNA, BPGM ACE 1201/4885REN 2613/4885LMNA 1077/4885
US-20130150416-A1 Glutamate receptor modulators and therapeutic agents GRM5, GRM1, GRIK5 ACE 2375/4885REN 1833/4885LMNA 4491/4885
US-20130324555-A1 Method of use of pharmaceutical formulations for the treatment of apicomplexan diseases in animals PIGS, ASAH2, ASAH1 ACE 219/4885REN 1746/4885LMNA 3632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.