SCHEMBL4270925

SCHEMBL4270925

CC(C)c1cc2c(cn1)OC1(CCNCC1)[C@H](C(=O)c1cc(-c3ccccc3)cc(-c3nnn[nH]3)c1)C2=O

nearest known ligand 0.30

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.30
OPRD1 P41143 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4267712 0.76 OPRD1 (0.32) CYP2D6OPRD1KCNH2
SCHEMBL4266728 0.76 OPRD1 (0.32) CYP2D6OPRD1KCNH2
SCHEMBL4266808 0.76 OPRD1 (0.32) CYP2D6OPRD1KCNH2
SCHEMBL731904 0.76 ACACB (0.44)
SCHEMBL4759175 0.72 ACACB (0.33)
SCHEMBL4411155 0.72 SCN9A (0.37) CYP2D6OPRD1KCNH2
SCHEMBL4275303 0.71 MAPT (0.30)
SCHEMBL4417848 0.70 KHK (0.38)
SCHEMBL4418928 0.70 ROCK2 (0.32)
SCHEMBL4270727 0.70 PIP5K1C (0.32) CYP2D6OPRD1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP claimed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO claimed
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed