SCHEMBL4275342

SCHEMBL4275342

CCCCc1ccc(-c2ccc(-c3ccc(OC(C(=O)O)c4ccccc4)cc3)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.64
RARB P10826 2/20 0.51
PPARA Q07869 8/20 0.49
PPARG P37231 7/20 0.49
FFAR1 O14842 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4529658 0.83 FFAR1 (0.47) PTPN1PPARAPPARGFFAR1
SCHEMBL4264241 0.80 PTPN1 (0.70) PTPN1
SCHEMBL17473054 0.79 RARB (0.58) RARBFFAR1
SCHEMBL7501649 0.79 PTPN1 (1.00) PTPN1
SCHEMBL11187778 0.77 CYP1A2 (0.56) PTPN1PPARAPPARG
SCHEMBL9472375 0.77 PPARG (0.60) PTPN1PPARAPPARGFFAR1
SCHEMBL14525686 0.77 FFAR1 (0.58) PTPN1RARBPPARAFFAR1
SCHEMBL4261546 0.77 SIRT3 (0.62) PTPN1
Bicarbonate SCHEMBL27623751 0.76 RARB (0.71) RARBFFAR1
SCHEMBL11756135 0.76 PTPN1 (0.51) PTPN1PPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090082392-A1 Substituted Carboxylic Acids THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY LLC 2009-03-26 US claimed
US-7358364-B2 treatment of diabetes and/or cancer; useful in the treatment of syndrome X; capable of inhibiting Protein tyrosine phosphatase THE INSTITUTE FOR PHARMACEUTICAL DISCOVERY LLC (US) 2008-04-15 US claimed
US-20040266788-A1 Substituted carboxylic acids THE INSTITUTE FOR PHARMACEUTICAL DISCOVERY LLC 2004-12-30 US claimed
US-20090082392-A1 Substituted Carboxylic Acids THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY LLC 2009-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040266788-A1 Substituted carboxylic acids PTP4A1, PTPRS, G6PC1 PTPN1 11/4885RARB 2880/4885PPARA 494/4885
US-20090082392-A1 Substituted Carboxylic Acids PTPRJ, PTPRS, PTPRG PTPN1 16/4885RARB 2640/4885PPARA 413/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.